SMARCA4/BRG1 Inhibitor Screening Assay Kit

32610

SMARCA2 Inhibitor Screening Assay Kit

The SMARCA2 Inhibitor Screening Assay Kit is designed to measure the inhibition of SMARCA2 binding to its substrate. The key to the SMARCA2 Inhibitor Screening Assay Kit is the specific binding of the SMARCA2 bromodomain to the acetylated histone substrate. With this kit, only three simple steps on a microtiter plate are required. First, a sample containing SMARCA2 and an inhibitor of choice is incubated with the biotinylated substrate for thirty minutes. Next, acceptor beads are added, then donor beads, followed by reading the Alpha-counts.

915 €

40341

SMARCA4/BRG1 TR-FRET Assay Kit

The SMARCA4 TR-FRET Assay Kit is designed to measure the inhibition of SMARCA4 binding to its substrate in a homogeneous 384 reaction format. This FRET-based assay requires no time-consuming washing steps, making it especially suitable for high throughput screening applications. The assay procedure is straightforward and simple; a sample containing terbium-labeled donor, dye-labeled acceptor, SMARCA4, substrate, and an inhibitor is incubated for 120 minutes. Then, the fluorescence intensity is measured using a fluorescence reader.

975 €

31102

SMARCA4 (BRG1), His-tag

Human BRG1, also known as SMARCA4, GenBank Accession No. NM_1128849, a.a. 1480 - 1603 corresponding to single bromodomain with N-terminal His-tag, MW = 15.5 kDa, expressed in an E. coli expression system.

607.5 €

HY-44012B

SMARCA-BD ligand 1 for Protac (hydrochloride)

SMARCA-BD ligand 1 hydrochloride for Protac is a compound that binds to the BAF ATPase subunits SMARCA2, and used for degrading SMARCA2, based on PROTAC[1].

1493.59 €

HY-44012A

SMARCA-BD ligand 1 for Protac (dihydrochloride)

SMARCA-BD ligand 1 for Protac dihydrochloride is a compound that binds to the BAF ATPase subunits SMARCA2, and used for degrading SMARCA2, based on PROTAC[1].

1493.59 €

MBS5754394-100mg

SMARCA-BD ligand 1 for Protac dihydrochloride

2467.25 €