HY-133126

hDDAH-1-IN-1

hDDAH-1-IN-1 (compound 8a) is a potent and selective non-amino acid catalytic site inhibitor of human dimethylarginine dimethylaminohydrolase-1 (hDDAH-1), with a Ki of 18 µM[1].

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HY-136300

PHD-1-IN-1

PHD-1-IN-1 is an orally active and potent HIF prolylhydroxylase domain-1 (PHD-1) inhibitor with an IC50 of 0.034 μM. PHD-1-IN-1 has a unique monodentate binding interaction with the active site Fe2+ ion and induces the formation of an “Arg367-out” pocket[1].

1849.57 €

HY-151891

TASK-1-IN-1

TASK-1-IN-1 is a potent and selective TASK-1 (Potassium Channel) inhibitor with an IC50 of 148 nM. TASK-1-IN-1 shows a reduced inhibition of TASK-3 channels (IC50 of 1750 nM) and not a significant effect on other K+ channels. TASK-1-IN-1 has anticancer effects.

787.09 €

MBS3844427-5x100mg

HO-1-IN-1

15813.69 €

MBS3611099-10mg

Enpp-1-IN-1

933.75 €

MBS3611099-25mg

Enpp-1-IN-1

1365.14 €