INT-777 (S-EMCA) is a potent and selective agonist of TGR5 receptor with EC50 value of 0.82 ?M [1]. TGR5 receptor is a G protein-coupled receptor and functions as a cell surface receptor for bile acids.
INT-777 (S-EMCA) is a potent and selective agonist of TGR5 receptor with EC50 value of 0.82 ?M [1]. TGR5 receptor is a G protein-coupled receptor and functions as a cell surface receptor for bile acids.