Dot1L-IN-1 (TFA)
5968.34 €
5968.34 €
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Catalog number: 804 - HY-101520A
Product Category: Business & Industrial > Science & Laboratory
Supplier:
Gentaur
Size: 1 mg
HY-138843A
FTO-IN-1 (TFA)
FTO-IN-1 TFA is a fat mass and obesity-associated enzyme (FTO) inhibitor extracted from patent WO2018157843A1, compound 32, with an IC50 of <1 μM. FTO-IN-1 TFA can be used for the research of cancer[1].
655.91 €
HY-139840A
GCPII-IN-1 (TFA)
GCPII-IN-1 TFA is a glutamate carboxypeptidase II (GCPII, or PSMA) inhibitor scaffold with a Ki of 44.3 nM[1].
2426.73 €
HY-144318
CREB-IN-1 (TFA)
CREB-IN-1 TFA is a potent, orally active CREB inhibitor (IC50=0.18 µM). CREB-IN-1 TFA inhibits breast cancer cell growth[1].
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Dot1L-IN-1 TFA is a highly potent and selective Dot1L inhibitor with a Ki of 2 pM and an IC50 of <0.1 nM. Dot1L-IN-1 TFA potently suppresses H3K79 dimethylation (IC50=3 nM), as well as the activity of the HoxA9 promoter (IC50=17 nM) in HeLa and Molm-13 cells, respectively[1].